MS094 2μM R03 exp136
Mechanism of Action
Inactive control for MS023 PRMT1 inhibitor
- Class / Subclass 1: Gene Regulation / Epigenetic Inhibitor
Technical Notes
Compound References
- PubChem Name: N/A
- Synonyms: N/A
- CAS #: 1831110-55-4
- PubChem CID: N/A
- IUPAC: N/A
- INCHI Name: N/A
- INCHI Key: N/A
- Molecular Weight: 288.2
- Canonical SMILES: N/A
- Isomeric SMILES: N/A
- Molecular Formula: C17H24N2O2
Compound Supplier
- Supplier Name: Structural Genomics Consortium
- Catalog #: N/A
- Lot #: N/A
Compound Characterization
- HRMS (ESI-TOF) m/z: (M+H)+ Calcd for C17H24N2O2 289.19105; found 289.19184
Dose Response Curve
- Platform ID: MS094
- Min: -7.1739; Max: 27.9782
| IC | Concentration (µM) |
|---|---|
| IC10 | N/A |
| IC20 | N/A |
| IC30 | N/A |
| IC40 | N/A |
| IC50 | N/A |
| IC60 | N/A |
| IC70 | N/A |
| IC80 | N/A |
| IC90 | N/A |
Screen Summary
- Round: 03
- Dose: 2µM
- Days of incubation: 8
- Doublings: 8.1
- Numbers of reads: 9689785
Screen Results
| Sensitive/Resistant hits (FDR<0.05) | CRANKS | Score Plot | Top 30 Genes | Screen Similarity | Top 30 Sensitive GO terms | Top 30 Resistant GO terms |
|---|---|---|---|---|---|---|
| 0/0 | Scores |